Rapamycin reverses chronic graft vascular disease in a novel cardiac allograft model

Circulation. 1999 Jul 6;100(1):67-74. doi: 10.1161/01.cir.100.1.67.

Abstract

Background: Chronic graft vascular disease (CGVD) in cardiac allografts has been defined as a slowly evolving vasculopathy unresponsive to conventional immunosuppression. We compared 4 rodent models of CGVD to evaluate the reproducibility of CGVD in heart allografts. Rapamycin (Rapa) and cyclosporine (CSA) were then used to treat CGVD.

Methods and results: Hearts were harvested and placed heterotopically into allogenic recipients. CGVD scores of PVG allografts from ACI recipients treated with CSA on days 1 through 10 were significantly elevated on day 90 (n=16) compared with other models (immunosuppression used): (1) Lewis to F344 recipients (CSA), (2) Brown Norway to Lewis (FK506), and (3) DA to Wistar-Firth (methylprednisolone, azathioprine, CSA). Although delayed (day 60 to 90) CSA treatment had no effect (n=6), delayed Rapa (3 mg. kg-1. d-1 IP) reversed CGVD in PVG grafts (0.22+/-0.19 on day 90, n=6). ACI isografts showed no evidence of CGVD (n=6) at day 90. Immunohistochemistry of PVG grafts revealed perivascular infiltrates consisting of CD4(+) T cells and limited numbers of macrophages persisting up to day 90. Flow cytometry demonstrated increased levels of anti-donor antibody at day 90, which was significantly inhibited by Rapa treatment.

Conclusions: PVG grafts developed a significant increase in CGVD without evidence of ongoing myocardial rejection. This CGVD appeared to be mediated by both cellular and humoral mechanisms, given CD4(+) perivascular infiltrates and increased levels of anti-donor antibody. The anti-CGVD effectiveness of Rapa during a period in which there was little myocardial cellular infiltrate supports a novel mechanism of effect such as smooth muscle or B-cell inhibition.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibody Formation / drug effects
  • Antibody Specificity
  • Coronary Disease / drug therapy*
  • Coronary Disease / etiology
  • Coronary Disease / immunology
  • Cyclosporine / therapeutic use
  • Drug Evaluation, Preclinical
  • Flow Cytometry
  • Graft Rejection
  • Graft vs Host Disease / drug therapy*
  • Graft vs Host Disease / etiology
  • Heart Transplantation / adverse effects*
  • Heart Transplantation / immunology
  • Histocompatibility
  • Histocompatibility Antigens / immunology
  • Immunity, Cellular / drug effects
  • Immunoglobulin G / blood
  • Immunosuppressive Agents / therapeutic use*
  • Isoantibodies / blood
  • Male
  • Nitric Oxide / physiology
  • Rats
  • Rats, Inbred ACI
  • Rats, Inbred F344
  • Rats, Inbred Lew
  • Rats, Inbred WF
  • Reproducibility of Results
  • Sirolimus / therapeutic use*
  • Transplantation, Homologous / adverse effects
  • Transplantation, Homologous / immunology

Substances

  • Histocompatibility Antigens
  • Immunoglobulin G
  • Immunosuppressive Agents
  • Isoantibodies
  • histocompatibility antigens RT, rat
  • Nitric Oxide
  • Cyclosporine
  • Sirolimus