Antimutagenic effect of plant flavonoids in the Salmonella assay system

Arch Pharm Res. 1994 Apr;17(2):71-5. doi: 10.1007/BF02974226.

Abstract

The antimutagenic effects of 27 kinds of plant flavonoids on the mutagenicity of aflatoxin B1(AFB1) and N-methyl-N'-nitro-N-nitrosoguanidine(MNNG) in Salmonella typhimurium TA100 were investigated. In the mixed applications of AFB1 (1 microgram/plate) with the flavonoids (300 micrograms/plate) in the presence of a mammalian metabolic activation system (S9 mix), chrysin, apigenin, luteolin and its glucoside, kaempferol, fisetin, morin, naringenin, hesperetin, persicogenin, (+)-catechin and (-)-epicatechin showed the antimutagenic effect against AFB1 with more than 70% inhibition rate. A little or no antimutagenicities except flavone against MNNG (0.5 microgram/plate) were observed. For the antimutagenicity of the flavonoids on AFB1, the flavonoid structure that contains the free 5-, 7-hydroxyl group seemed to be essential. However, saturation of the 2,3-double bond or elimination of the 4-keto group did not affect the activity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aflatoxin B1 / toxicity
  • Animals
  • Antimutagenic Agents / isolation & purification
  • Antimutagenic Agents / pharmacology*
  • Antimutagenic Agents / toxicity
  • Catechin / pharmacology
  • Flavonoids / isolation & purification
  • Flavonoids / pharmacology*
  • Flavonoids / toxicity
  • In Vitro Techniques
  • Methylnitronitrosoguanidine / toxicity
  • Mutagenicity Tests
  • Mutagens / toxicity
  • Rats
  • Salmonella typhimurium / drug effects*
  • Salmonella typhimurium / genetics

Substances

  • Antimutagenic Agents
  • Flavonoids
  • Mutagens
  • Methylnitronitrosoguanidine
  • Catechin
  • Aflatoxin B1