A contraceptive peptide vaccine targeting sulfated glycoprotein ZP2 of the mouse zona pellucida

Biol Reprod. 1999 Apr;60(4):900-7. doi: 10.1095/biolreprod60.4.900.

Abstract

In this study, we have mapped and characterized a B cell epitope of sulfated glycoprotein ZP2 (ZP2) as a step toward the development of a multi-epitope zona pellucida (ZP) vaccine. Recombinant polypeptides expressed by random deoxyribonuclease-digested fragments of ZP2 cDNA were screened for binding to IE-3, a monoclonal antibody to murine ZP2. Positive clones contained cDNA inserts encoding polypeptide corresponding to ZP2(103-134). When normal or ovariectomized female mice were immunized with three overlapping peptides that span this region of ZP2 (101-120, 111-130, 121-140), only ZP2(121-140) elicited IgG antibodies that reacted with mouse ovarian ZP, indicative of the presence of native B epitope and helper T cell epitope in ZP2(121-140). To more finely map the ZP2 B cell epitope, a random peptide display library was screened with the IE-3 antibody, and a consensus tetramer sequence VxYK that matched the ZP2(123-126) sequence VRYK was located. Competitive immunofluorescence analysis with single alanine-substituted VxYK peptides ranked the relative contribution of the three critical B cell epitope residues as Y > V > K. A chimeric peptide was constructed that contained the YRYK motif of ZP2 and a bovine RNase T cell epitope. Although (C57BL/6xA/J) F1 (B6AF1) female mice immunized with the chimeric peptide developed ZP antibody response, this peptide elicited antibody only in mice of the histocompatibility complex (MHC) H-2(k or b) haplotype. In contrast, ZP2(121-140) peptide elicited antibody in inbred mice with three additional mouse MHC haplotypes. Moreover, although ZP2(121-140) contained a T cell epitope, no oophoritis was observed after immunization of B6AF1 mice with ZP2(121-140) in complete Freund's adjuvant (CFA). In a preliminary trial, female B6AF1 mice immunized with ZP2(121-140) in CFA had reduced litter sizes as compared with mice injected with CFA alone.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Contraception, Immunologic*
  • Egg Proteins / chemistry
  • Egg Proteins / immunology*
  • Epitope Mapping
  • Epitopes / chemistry
  • Epitopes / immunology
  • Female
  • Immunoglobulin G / immunology
  • Male
  • Membrane Glycoproteins / chemistry
  • Membrane Glycoproteins / immunology*
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred C3H
  • Mice, Inbred C57BL
  • Mice, Inbred DBA
  • Molecular Sequence Data
  • Ovariectomy
  • Receptors, Cell Surface*
  • Recombinant Fusion Proteins / immunology
  • T-Lymphocytes, Helper-Inducer / immunology
  • Vaccines*
  • Zona Pellucida / immunology
  • Zona Pellucida Glycoproteins

Substances

  • Egg Proteins
  • Epitopes
  • Immunoglobulin G
  • Membrane Glycoproteins
  • Receptors, Cell Surface
  • Recombinant Fusion Proteins
  • Vaccines
  • Zona Pellucida Glycoproteins
  • Zp2 protein, mouse