Evaluation of topical application of clobetasol 17-propionate from various cream bases

Drug Dev Ind Pharm. 1999 Jan;25(1):7-14. doi: 10.1081/ddc-100102136.

Abstract

The effect of clobetasol 17-propionate (CP), a potent corticosteroid, in various cream bases on the permeation through artificial membrane was sought. Four formulations were then chosen for a further in vivo skin blanching assay. After calculation of the relationship between in vivo flux0-8 hr determined from a surface recovery technique and in vitro release rate0-8 hr of CP from various formulations, a high correlation coefficient of 0.9996 was achieved. Therefore, the in vitro release study could be used as an index to predict and evaluate the in vivo penetration capacity of CP cream to screen the effective formulation preclinically. After a series of in vivo investigations in this study, it was concluded that myristic acid-added formulations may show a bioequivalence with commercial Dermovate. Furthermore, the flux calculated from the surface recovery technique and delta E detected from the skin blanching assay may be useful as parameters evaluating the quality and effectiveness of CP cream.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Topical
  • Adult
  • Anti-Inflammatory Agents / administration & dosage
  • Anti-Inflammatory Agents / pharmacokinetics*
  • Chemistry, Pharmaceutical / methods
  • Chromatography, High Pressure Liquid
  • Clobetasol / administration & dosage
  • Clobetasol / analogs & derivatives*
  • Clobetasol / pharmacokinetics
  • Colorimetry
  • Glucocorticoids
  • Humans
  • Male
  • Membranes, Artificial
  • Myristic Acid
  • Ointment Bases
  • Ointments
  • Skin / blood supply
  • Skin / drug effects
  • Therapeutic Equivalency
  • Time Factors
  • Vasoconstriction / drug effects
  • Viscosity

Substances

  • Anti-Inflammatory Agents
  • Glucocorticoids
  • Membranes, Artificial
  • Ointment Bases
  • Ointments
  • Myristic Acid
  • Clobetasol